KEGG   DRUG: Etokimab
Entry
D11449                      Drug                                   
Name
Etokimab (USAN)
Formula
C6534H10088N1724O2018S46
Exact mass
146464.6915
Mol weight
146555.3425
Sequence
(Heavy chain)
QVQLMQSGAE VKKPGASVKV SCKASGYTFT SYWMHWVRQA PGQGLEWMGT IYPRNSNTDY
NQKFKARVTM TRDTSTSTVY MELSSLRSED TAVYYCARPL YYYLTSPPTL FWGQGTLVTV
SSASTKGPSV FPLAPSSKST SGGTAALGCL VKDYFPEPVT VSWNSGALTS GVHTFPAVLQ
SSGLYSLSSV VTVPSSSLGT QTYICNVNHK PSNTKVDKKV EPKSCDKTHT CPPCPAPELL
GGPSVFLFPP KPKDTLMISR TPEVTCVVVD VSHEDPEVKF NWYVDGVEVH NAKTKPREEQ
YNSTYRVVSV LTVLHQDWLN GKEYKCKVSN KALPAPIEKT ISKAKGQPRE PQVYTLPPSR
DELTKNQVSL TCLVKGFYPS DIAVEWESNG QPENNYKTTP PVLDSDGSFF LYSKLTVDKS
RWQQGNVFSC SVMHEALHNH YTQKSLSLSP GK
(Light chain)
DIQLTQSPSF LSASVGDRVT ITCKASQDVG TAVAWYQQKP GKAPKLLIYW ASTRHTGVPS
RFSGSGSGTE FTLTISSLQP EDFATYYCQQ AKTYPFTFGS GTKLEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H149-H205, H225-L214, H231-H'231, H234-H'234, H266-H326, H372-H430, H'22-H'96, H'149-H'205, H'225-L'214, H'266-H'326, H'372-H'430, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Class
Immunological agent
 DG02019  Interleukin inhibitor
Efficacy
Anti-inflammatory, Anti-interleukin 33 antibody
  Type
Monoclonal antibody
Comment
Treatment of patients with peanut allergy, dermatitis, and asthma
Target
IL33 [HSA:90865] [KO:K12967]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04217  Necroptosis
hsa04623  Cytosolic DNA-sensing pathway
Brite
Drug groups [BR:br08330]
 Immunological agent
  DG02019  Interleukin inhibitor
   D11449  Etokimab
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Interleukins
    IL33
     D11449  Etokimab (USAN)
Other DBs
CAS: 2022981-44-6
PubChem: 384585426
LinkDB

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