KEGG   DRUG: Dilpacimab
Entry
D11642                      Drug                                   
Name
Dilpacimab (USAN/INN)
Formula
C8888H13570N2342O2768S58
Exact mass
199255.6888
Mol weight
199378.648
Sequence
(Heavy chain)
EVQLVESGGG LVQPGGSLRL SCAASGFTFS NFPMAWVRQA PGKGLEWVAT ISSSDGTTYY
RDSVKGRFTI SRDNAKNSLY LQMNSLRAED TAVYYCARGY YNSPFAYWGQ GTLVTVSSAS
TKGPEVQLVE SGGGLVQPGG SLRLSCAASG YTFTNYGMNW VRQAPGKGLE WVGWINTYTG
EPTYAADFKR RFTFSLDTSK STAYLQMNSL RAEDTAVYYC AKYPHYYGSS HWYFDVWGQG
TLVTVSSAST KGPSVFPLAP SSKSTSGGTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF
PAVLQSSGLY SLSSVVTVPS SSLGTQTYIC NVNHKPSNTK VDKKVEPKSC DKTHTCPPCP
APEAAGGPSV FLFPPKPKDT LMISRTPEVT CVVVDVSHED PEVKFNWYVD GVEVHNAKTK
PREEQYNSTY RVVSVLTVLH QDWLNGKEYK CKVSNKALPA PIEKTISKAK GQPREPQVYT
LPPSREEMTK NQVSLTCLVK GFYPSDIAVE WESNGQPENN YKTTPPVLDS DGSFFLYSKL
TVDKSRWQQG NVFSCSVMHE ALHNHYTQKS LSLSPGK
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRASEDIY SNLAWYQQKP GKAPKLLIYD
TNNLADGVPS RFSGSGSGTD FTLTISSLQP EDFATYYCQQ YNNYPPTFGQ
GTKLEIKRTV AAPSVFIFPP DIQMTQSPSS LSASVGDRVT ITCSASQDIS NYLNWYQQKP
GKAPKVLIYF TSSLHSGVPS RFSGSGSGTD FTLTISSLQP EDFATYYCQQ YSTVPWTFGQ
GTKVEIKRTV AAPSVFIFPP SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ
ESVTEQDSKD STYSLSSTLT LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H146-H220, H274-H330, H350-L334, H356-H'356, H359-H'359, H391-H451, H497-H555, H'22-H'96, H'146-H'220, H'274-H'330, H'350-L'334, H'391-H'451, H'497-H'555, L23-L88, L143-L208, L254-L314, L'23-L'88, L'143-L'208, L'254-L'314)
  Type
Peptide
Efficacy
Antineoplastic
  Type
Monoclonal antibody, bispecific antibody
Target
DLL4 [HSA:54567] [KO:K06051]
VEGFA [HSA:7422] [KO:K05448]
  Pathway
hsa04014  Ras signaling pathway
hsa04151  PI3K-Akt signaling pathway
hsa04330  Notch signaling pathway
hsa04370  VEGF signaling pathway
hsa05200  Pathways in cancer
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Growth factors (RTK-binding)
    VEGFA
     D11642  Dilpacimab (USAN/INN)
 Not elsewhere classified
  Signaling molecules
   Notch signaling
    DLL4
     D11642  Dilpacimab (USAN/INN)
Other DBs
CAS: 1791420-09-1
PubChem: 405226509
LinkDB

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