KEGG   DRUG: Fletikumab
Entry
D11756                      Drug                                   
Name
Fletikumab (USAN/INN)
Formula
C6494H10000N1728O2050S44
Exact mass
146399.9083
Mol weight
146490.0934
Sequence
(Heavy chain)
QVQLVQSGAE VKRPGASVKV SCKASGYTFT NDIIHWVRQA PGQRLEWMGW INAGYGNTQY
SQNFQDRVSI TRDTSASTAY MELISLRSED TAVYYCAREP LWFGESSPHD YYGMDVWGQG
TTVTVSSAST KGPSVFPLAP CSRSTSESTA ALGCLVKDYF PEPVTVSWNS GALTSGVHTF
PAVLQSSGLY SLSSVVTVPS SSLGTKTYTC NVDHKPSNTK VDKRVESKYG PPCPPCPAPE
FLGGPSVFLF PPKPKDTLMI SRTPEVTCVV VDVSQEDPEV QFNWYVDGVE VHNAKTKPRE
EQFNSTYRVV SVLTVLHQDW LNGKEYKCKV SNKGLPSSIE KTISKAKGQP REPQVYTLPP
SQEEMTKNQV SLTCLVKGFY PSDIAVEWES NGQPENNYKT TPPVLDSDGS FFLYSRLTVD
KSRWQEGNVF SCSVMHEALH NHYTQKSLSL SLGK
(Light chain)
AIQLTQSPSS LSASVGDRVT ITCRASQGIS SALAWYQQKP GKAPKLLIYD ASSLESGVPS
RFSGSGSGTD FTLTISSLQP EDFATYYCQQ FNSYPLTFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG LSSPVTKSFN RGEC
(Disulfide bridge: H22-H96, H141-L214, H154-H210, H233-H'233, H236-H'236, H268-H328, H374-H432, H'22-H'96, H'141-L'214, H'154-H'210 H'268-H'328, H'374-H'432, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Antirheumatic, Anti-IL-20 antibody
  Type
Monoclonal antibody
Comment
Treatment of rheumatoid arthritis
Target
IL20 [HSA:50604] [KO:K22667]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04630  JAK-STAT signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Interleukins
    IL20
     D11756  Fletikumab (USAN/INN)
Other DBs
CAS: 1357158-22-5
PubChem: 405226622
LinkDB

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