KEGG   DRUG: Dazukibart
Entry
D12464                      Drug                                   
Name
Dazukibart (USAN)
Formula
C6472H9998N1716O2017S46
Exact mass
145501.9677
Mol weight
145591.9115
Sequence
(Heavy chain)
QVQLVQSGAE VKKPGSSVKV SCKASGYTFS RYWMHWVRQA PGQGLEWMGH IDPSDSYTYY
NQKFKGRVTI TADESTSTAY MELSSLRSED TAVYYCARWD YGNLLFEYWG QGTLVTVSSA
STKGPSVFPL APSSKSTSGG TAALGCLVKD YFPEPVTVSW NSGALTSGVH TFPAVLQSSG
LYSLSSVVTV PSSSLGTQTY ICNVNHKPSN TKVDKKVEPK SCDKTHTCPP CPAPEAAGAP
SVFLFPPKPK DTLMISRTPE VTCVVVDVSH EDPEVKFNWY VDGVEVHNAK TKPREEQYNS
TYRVVSVLTV LHQDWLNGKE YKCKVSNKAL PAPIEKTISK AKGQPREPQV YTLPPSREEM
TKNQVSLTCL VKGFYPSDIA VEWESNGQPE NNYKTTPPVL DSDGSFFLYS KLTVDKSRWQ
QGNVFSCSVM HEALHNHYTQ KSLSLSPG
(Light chain)
DIQMTQSPSS LSASVGDRVT ITCRTSQDIG NYLNWYQQKP GKAFKLLIYS TSRLHSGVPS
RFSGSGSGTD FTLTISSLQP EDFATYYCQQ GIILPITFGG GTKVEIKRTV AAPSVFIFPP
SDEQLKSGTA SVVCLLNNFY PREAKVQWKV DNALQSGNSQ ESVTEQDSKD STYSLSSTLT
LSKADYEKHK VYACEVTHQG
(Disulfide bridge: H22-H96, H146-H202, H222-L214, H228-H'228, H231-H'231, H263-H323, H369-H427, H'22-H'96, H'146-H'202, H'222-L'214, H'263-H'323, H'369-H'427, L23-L88, L134-L194, L'23-L'88, L'134-L'194)
  Type
Peptide
Efficacy
Anti-inflammatory disease
  Type
Monoclonal antibody
Comment
Treatment of dermatomyositis and systemic lupus erythematosus
Target
IFNB [HSA:3456] [KO:K05415]
  Pathway
hsa04060  Cytokine-cytokine receptor interaction
hsa04620  Toll-like receptor signaling pathway
hsa04621  NOD-like receptor signaling pathway
hsa04668  TNF signaling pathway
Brite
Target-based classification of drugs [BR:br08310]
 Cytokines and receptors
  Cytokines
   Interferons
    IFNB
     D12464  Dazukibart (USAN)
Other DBs
CAS: 2639474-65-8
LinkDB

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