| beta1-Adrenergic receptor antagonist |
| Practolol (USAN) |
| Metoprolol |
| Metoprolol (USAN/INN) |
| Metoprolol tartrate (JP18/USP) <JP/US> |
| Metoprolol succinate (USP) <US> |
| Metoprolol fumarate (USP) |
| Atenolol (JP18/USP/INN) <JP/US> |
| Acebutolol |
| Acebutolol (USAN/INN) |
| Acebutolol hydrochloride (JP18/USP) <US> |
| Betaxolol |
| Betaxolol (INN) |
| Betaxolol hydrochloride (JP18/USP) <JP/US> |
| Bisoprolol |
| Bisoprolol (JAN/USAN/INN) <JP> |
| Bisoprolol fumarate (JP18/USP) <JP/US> |
| Celiprolol |
| Celiprolol (INN) |
| Celiprolol hydrochloride (JAN/USAN) <JP> |
| Esmolol |
| Esmolol (INN) |
| Esmolol hydrochloride (JAN/USP) <JP/US> |
| Epanolol (USAN/INN) |
| Esatenolol (JAN/INN) |
| Nebivolol |
| Nebivolol (USAN/INN) |
| Nebivolol hydrochloride (USAN) <US> |
| Talinolol (INN) |
| Landiolol |
| Landiolol (USAN/INN) |
| Landiolol hydrochloride (JAN/USAN) <JP> |
| Cetamolol hydrochloride (USAN) |
| Cicloprolol hydrochloride (USAN) |
| Levobetaxolol hydrochloride (USAN) |
| beta2-Adrenergic receptor antagonist |
| Bucindolol hydrochloride (USAN) |
| Butoxamine hydrochloride (USAN) |
| Carazolol (INN) |
| Alprenolol |
| Alprenolol (INN) |
| Alprenolol hydrochloride (JP18/USAN) |
| Oxprenolol |
| Oxprenolol (INN) |
| Oxprenolol hydrochloride (JP18/USP) |
| Pindolol (JP18/USP/INN) <JP/US> |
| Propranolol |
| Propranolol (INN) |
| Propranolol hydrochloride (JP18/USP) <JP/US> |
| Timolol |
| Timolol (INN) |
| Timolol (USAN) <US> |
| Timolol maleate (JP18/USP) <JP/US> |
| Sotalol |
| Sotalol (INN) |
| Sotalol hydrochloride (JAN/USP) <JP/US> |
| Nadolol (JP18/USP/INN) <JP/US> |
| Mepindolol (INN) |
| Carteolol |
| Carteolol (INN) |
| Carteolol hydrochloride (JP18/USP) <JP/US> |
| Tertatolol |
| Tertatolol (INN) |
| Tertatolol hydrochloride |
| Bopindolol |
| Bopindolol (INN) |
| Bopindolol malonate (JAN) |
| Bupranolol |
| Bupranolol (INN) |
| Bupranolol hydrochloride (JP18) |
| Penbutolol |
| Penbutolol (INN) |
| Penbutolol sulfate (JP18/USP) |
| Cloranolol (INN) |
| Levobunolol |
| Levobunolol (INN) |
| Levobunolol hydrochloride (JAN/USP) <JP/US> |
| Metipranolol |
| Metipranolol (USAN/INN) |
| Metipranolol hydrochloride |
| Befunolol |
| Befunolol (INN) |
| Befunolol hydrochloride (JAN) |
| Bufetolol hydrochloride (JP18) <JP> |
| Medroxalol |
| Medroxalol (USAN/INN) |
| Medroxalol hydrochloride (USAN) |
| Tilisolol |
| Tilisolol (INN) |
| Tilisolol hydrochloride (JAN) |
| Indenolol |
| Indenolol (INN) |
| Indenolol hydrochloride (JP18) |
| Bucumolol hydrochloride (JP18) |
| Primidolol (USAN/INN) |
| Adaprolol maleate (USAN) |
| Alprenoxime hydrochloride (USAN) |
| Bunolol hydrochloride (USAN) |
| Dexpropranolol hydrochloride (USAN) |
| Diacetolol hydrochloride (USAN) |
| Flestolol sulfate (USAN) |
| Pamatolol sulfate (USAN) |
| Beradilol monoethyl maleate (JAN) |